Cholestyramine is a cholesterol-lowering drug that belongs to thebile acid resin classof medications, also called bile acid sequestrants.
Cholestyramine has also been shown to slow the progression of the development of atherosclerosis in a couple of studies.
However, it has not been shown to prevent death or disability due to cardiovascular disease.
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How Does Cholestyramine Work?
When cholestyramine binds to bile acids, they become depleted and will not be reabsorbed.
To make more bile acids, cholesterol will be removed from the bloodstream and converted into bile acids.
This activity lowers your cholesterol levels.
How Should You Take Cholestyramine?
You should take cholestyramine as directed by your healthcare provider.
Cholestyramine is available in a powdered form, packaged into small, single-dose packets or in a larger container.
You should ingest the entire contents of the drink containing cholestyramine to get the full dose of the medication.
Cholestyramine should be taken with a meal.
Who Shouldnt Take It?
Due to its components, there are some instances where cholestyramine should not be taken.
This usually goes away with continued treatment.
Other common side effects include:
Other side effects have been reported due to prolonged use of cholestyramine.
Prolonged drinking of the product or holding the product in the mouth may cause tooth enamel erosion or discoloration.
This will help your healthcare provider to identify any potential interactions between cholestyramine and your other medications.
Bottom Line
Cholestyramine is one of the first cholesterol-lowering medications approved in the United States.
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